nazwa: JB170
nr katalogowy: GC63707-10
cas: 2705844-82-0
producent: GLPBio
opakowanie: 10mg
cena: 3784,46 [Pln] (bez rabatu)
wyszukaj podobne produkty: 2705844-82-0
Formula: C48H44ClFN8O11. Molecular weight: 963,36. Solubility: DMSO : 100 mg/mL (103.80 mM, Need ultrasonic). Storage: Store at -20°C. Synonym: JB170 is a potent and highly specific PROTAC-mediated AURORA-A (Aurora Kinase) degrader (DC50=28 nM) by linking Alisertib, to the Cereblon-binding molecule Thalidomide. JB170 preferentially binds AURORA-A (EC50=193 nM) over AURORA-B (EC50=1.4 ?M). JB170-mediated S-phase arrest is caused specifically by AURORA-A depletion. JB170 has excellent ability to inhibit non-catalytic function of AURORA-A kinase..
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czas dostawy: Do potwierdzenia przez Chemat