RLX–33 cas: (2784577-71-3)

nazwa: RLX–33

nr katalogowy: GC69821-1

cas: 2784577-71-3

producent: GLPBio

opakowanie: 1mg

cena: 1046,37 [Pln] (bez rabatu)

wyszukaj podobne produkty: 2784577-71-3


szczegóły:

Formula: C24H19ClN4O4. Molecular weight: 462,89. Solubility: DMSO : 125 mg/mL (270.04 mM, Need ultrasonic). Storage: Store at -20°C. Synonym: RLX-33 is an effective and selective relaxin family peptide 3 (RXFP3) antagonist with blood-brain barrier permeability. It also blocks the phosphorylation of ERK1/2 induced by relaxin 3, with IC50 values for RXFP3, ERK1, and ERK2 phosphorylation being 2.36 μM, 7.82 μM, and 13.86 μM respectively. RLX-33 can block the increase in food intake induced by the RXFP3 selective agonist R3/I5 in rats. RLX-33 can be used for research on metabolic syndrome..

właściwości

czystość: No data

czas dostawy: Do potwierdzenia przez Chemat