nazwa: TAK–243 (MLN7243)
nr katalogowy: GC32737-5
cas: 1450833-55-2
producent: GLPBio
opakowanie: 5mg
cena: 1139,98 [Pln] (bez rabatu)
wyszukaj podobne produkty: 1450833-55-2
Formula: C19H20F3N5O5S2. Molecular weight: 519,52. Solubility: DMSO : 50 mg/mL (96.24 mM),Water : 1 mg/mL (1.92 mM). Storage: Store at -20°C. Synonym: TAK-243 (MLN7243) (MLN7243) is a first-in-class, selective ubiquitin activating enzyme, UAE (UBA1) inhibitor (IC50=1 nM), which blocks ubiquitin conjugation, disrupting monoubiquitin signaling as well as global protein ubiquitination. TAK-243 (MLN7243) (MLN7243) induces endoplasmic reticulum (ER) stress, abrogates NF-κB pathway activation and promotes apoptosis..
czystość: No data
czas dostawy: Do potwierdzenia przez Chemat