nazwa: Tazemetostat hydrobromide
nr katalogowy: GC38163-100
cas: 1467052-75-0
producent: GLPBio
opakowanie: 100mg
cena: 1930,98 [Pln] (bez rabatu)
wyszukaj podobne produkty: 1467052-75-0
Formula: C34H45BrN4O4. Molecular weight: 653,65. Solubility: DMSO: 100 mg/mL (152.99 mM). Storage: Store at -20°C. Synonym: Tazemetostat hydrobromide (EPZ-6438 hydrobromide) is a potent, selective and orally available EZH2 inhibitor. Tazemetostat hydrobromide inhibits the activity of human polycomb repressive complex 2 (PRC2)-containing wild-type EZH2 with a Ki value of 2.5 nM. Tazemetostat hydrobromide inhibits EZH2 with IC50s of 11 and 16 nM in peptide assay and nucleosome assay, respectively. Tazemetostat hydrobromide inhibits Rat EZH2 with an IC50 of 4 nM. Tazemetostat hydrobromide also inhibits EZH1 with an IC50 of 392 nM..
czystość: No data
czas dostawy: Do potwierdzenia przez Chemat