nazwa: Samuraciclib hydrochloride hydrate
nr katalogowy: GC63736-5
producent: GLPBio
opakowanie: 5mg
cena: 1233,59 [Pln] (bez rabatu)
wyszukaj podobne produkty: GC63736-5
Formula: C22H30N6O.(2.5HCl).(2H2O). Molecular weight: 521,7. Solubility: DMSO : 100 mg/mL (191.68 mM, Need ultrasonic). Storage: 4°C, stored under nitrogen, away from moisture. Synonym: Samuraciclib (CT7001) hydrochloride hydrate is a potent, selective, ATP-competitive and orally active CDK7 inhibitor, with an IC50 of 41 nM. Samuraciclib hydrochloride hydrate displays 45-, 15-, 230- and 30-fold selectivity over CDK1, CDK2 (IC50 of 578 nM), CDK5 and CDK9, respectively. Samuraciclib hydrochloride hydrate inhibits the growth of breast cancer cell lines with GI50 values between 0.2-0.3 ?M. Samuraciclib hydrochloride hydrate has anti-tumor effects..
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czas dostawy: Do potwierdzenia przez Chemat