GSK1016790A

cas: 942206-85-1 — see every product listed under this CAS number, including other names

GSK1016790A (CAS 942206-85-1) is a chemical reagent available from Chemat. Available pack sizes: 10mg, 25mg, 5mg, 50mg, 100mg. Offered by: GLPBio, Biosynth, Sigma-Aldrich.

brandGLPBio
catalog numberGC17940-10
cas942206-85-1
size10mg
Need more information?

Ask us about this product — we're happy to help.

Available pack sizes

brand size price
GLPBio 10mg 779.58 Pln
GLPBio 25mg 1177.42 Pln
GLPBio 5mg 657.89 Pln
Biosynth 25mg price on request
Biosynth 50mg price on request
Biosynth 100mg price on request
Sigma-Aldrich 10MG 1250.00 Pln
Sigma-Aldrich 50MG 4880.00 Pln

properties

purityNo data
delivery timeTo be confirmed by Chemat
Structural formula: {0} (CAS {1})

GSK1016790A is a tertiary carboxamide that is piperazine in which one of the amino groups has undergone condensation with the carboxy group of N-[(2,4-dichlorophenyl)sulfonyl]-L-serine, while the other has undergone condensation with the carboxy group of N-(1-benzothiophen-2-ylcarbonyl)-L-leucine. It is a cell-permeable, potent and selective agonist of the TRPV4 (transient receptor potential vanilloid 4) channel. It has a role as a TRPV4 agonist. It is a tertiary carboxamide, a dichlorobenzene, an aromatic primary alcohol, a sulfonamide, a member of 1-benzothiophenes and a N-acylpiperazine.

Source: ChEBI

Identity
Molecular formulaC28H32Cl2N4O6S2
Molecular weight655.6 g/mol
IUPAC nameN-[(2S)-1-[4-[(2S)-2-[(2,4-dichlorophenyl)sulfonylamino]-3-hydroxypropanoyl]piperazin-1-yl]-4-methyl-1-oxopentan-2-yl]-1-benzothiophene-2-carboxamide
InChIKeyIVYQPSHHYIAUFO-VXKWHMMOSA-N
SMILESCC(C)C[C@@H](C(=O)N1CCN(CC1)C(=O)[C@H](CO)NS(=O)(=O)C2=C(C=C(C=C2)Cl)Cl)NC(=O)C3=CC4=CC=CC=C4S3

Computed by PubChem (NCBI)

Also listed as