Lorlatinib

cas: 1454846-35-5 — see every product listed under this CAS number, including other names

Lorlatinib (CAS 1454846-35-5) is a chemical reagent available from Chemat. Available pack sizes: 0,05g, 0,1g, 0,25g, 0,5g, 1g. Offered by: Biosynth.

brandBiosynth
catalog numberFP104236-0,05g
cas1454846-35-5
size0,05g
Need more information?

Ask us about this product — we're happy to help.

Available pack sizes

brand size price
Biosynth 0,05g price on request
Biosynth 0,1g price on request
Biosynth 0,25g price on request
Biosynth 0,5g price on request
Biosynth 1g price on request

properties

categoryLife Sciences
sub-category 1Ligands
sub-category 2Enzyme Modulators
purityNo data
delivery time1-2 weeks

Lorlatinib is a cyclic ether that is 16,17-dihydro-2H-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10H)-one substituted by methyl groups at positions 2 and 10R, and by cyano, amino and fluoro groups at positions 3, 7 and 12 respectively. It is a small molecule inhibitor of ALK and ROS1 kinase developed by Pfizer for the treatment of ALK-positive non-small cell lung cancer. It has a role as an antineoplastic agent and an EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor. It is a nitrile, a member of benzamides, a member of pyrazoles, an aromatic ether, a cyclic ether, an organic heterotetracyclic compound, an aminopyridine, an azamacrocycle and a member of monofluorobenzenes.

Source: ChEBI

Identity
Molecular formulaC21H19FN6O2
Molecular weight406.4 g/mol
IUPAC name(16R)-19-amino-13-fluoro-4,8,16-trimethyl-9-oxo-17-oxa-4,5,8,20-tetrazatetracyclo[16.3.1.02,6.010,15]docosa-1(22),2,5,10(15),11,13,18,20-octaene-3-carbonitrile
InChIKeyIIXWYSCJSQVBQM-LLVKDONJSA-N
SMILESC[C@@H]1C2=C(C=CC(=C2)F)C(=O)N(CC3=NN(C(=C3C4=CC(=C(N=C4)N)O1)C#N)C)C

Computed by PubChem (NCBI)

Also listed as