SKF 83822 hydrobromide
cas: 74115-10-9 — see every product listed under this CAS number, including other names
SKF 83822 hydrobromide (CAS 74115-10-9) is a chemical reagent available from Chemat. Available pack sizes: 10mg, 50mg. Offered by: GLPBio.
| brand | GLPBio |
|---|---|
| catalog number | GC11503-10 |
| cas | 74115-10-9 |
| size | 10mg |
Need more information?
Ask us about this product — we're happy to help.
Available pack sizes
| brand | size | price | |
|---|---|---|---|
| GLPBio | 10mg | 1692.28 Pln | |
| GLPBio | 50mg | 5778.35 Pln |
properties
| purity | No data |
|---|---|
| delivery time | To be confirmed by Chemat |
N-allyl-6-chloro-1-(3-methylphenyl)-2,3,4,5-tetrahydro-3-benzazepine-7,8-diol hydrobromide is a hydrobromide salt prepared from N-allyl-6-chloro-1-(3-methylphenyl)-2,3,4,5-tetrahydro-3-benzazepine-7,8-diol and one equivalent of hydrogen bromide. High affinity, selective dopamine D1-like receptor agonist. Ki values are 3.2, 3.1, 186, 66, 335, 1167, 1251 and 1385 nM at recombinant D1, D5, D2, D3, D4, 5-HT2A, alpha1A and alpha1B receptors respectively. Stimulates adenylyl cyclase (EC50 = 65 nM) but not phosphoinositide hydrolysis. Induces extreme arousal and hyperlocomotion following subcutaneous administration in monkeys. It has a role as a prodrug and a dopamine agonist. It contains a N-allyl-6-chloro-1-(3-methylphenyl)-2,3,4,5-tetrahydro-3-benzazepinium-7,8-diol(1+).
Source: ChEBI
| Molecular formula | C20H23BrClNO2 |
|---|---|
| Molecular weight | 424.8 g/mol |
| IUPAC name | 9-chloro-5-(3-methylphenyl)-3-prop-2-enyl-1,2,4,5-tetrahydro-3-benzazepine-7,8-diol;hydrobromide |
| InChIKey | CFWPKYBBXBANLU-UHFFFAOYSA-N |
| SMILES | CC1=CC(=CC=C1)C2CN(CCC3=C(C(=C(C=C23)O)O)Cl)CC=C.Br |
Computed by PubChem (NCBI)
Synonyms:
orb1704058