Bictegravir

cas: 1611493-60-7 — see every product listed under this CAS number, including other names

Bictegravir (CAS 1611493-60-7) is a chemical reagent available from Chemat. Available pack sizes: on request, 50mg, 10mg. Offered by: Chemat Brand, Biosynth.

brandChemat Brand
catalog numberULB167001
cas1611493-60-7
sizeon request
availability Do potwierdzenia przez Chemat|To be confirmed by Chemat
Need more information?

Ask us about this product — we're happy to help.

Available pack sizes

brand size price
Chemat Brand on request price on request
Biosynth 50mg price on request
Biosynth 10mg price on request

properties

purityNo data
categoryChemicals
delivery timeTo be confirmed by Chemat

Bictegravir is a monocarboxylic acid amide obtained by formal condensation of the carboxy group of (2R,5S,13aR)-8-hydroxy-7,9-dioxo-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxylic acid with the amino group of 2,4,6-trifluorobenzylamine. It is a second-generation integrase strand transfer inhibitor (INSTI) and used (as its sodium salt) for the treatment of HIV-1. It has a role as a HIV-1 integrase inhibitor. It is a secondary carboxamide, a monocarboxylic acid amide, an organic heterotetracyclic compound and a trifluorobenzene. It is a conjugate acid of a bictegravir(1-).

Source: ChEBI

Identity
Molecular formulaC21H18F3N3O5
Molecular weight449.4 g/mol
IUPAC name(1S,11R,13R)-5-hydroxy-3,6-dioxo-N-[(2,4,6-trifluorophenyl)methyl]-12-oxa-2,9-diazatetracyclo[11.2.1.02,11.04,9]hexadeca-4,7-diene-7-carboxamide
InChIKeySOLUWJRYJLAZCX-LYOVBCGYSA-N
SMILESC1C[C@@H]2C[C@H]1N3[C@H](O2)CN4C=C(C(=O)C(=C4C3=O)O)C(=O)NCC5=C(C=C(C=C5F)F)F

Computed by PubChem (NCBI)

Also listed as