EPZ5676

cas: 1380288-87-8 — see every product listed under this CAS number, including other names

EPZ5676 (CAS 1380288-87-8) is a chemical reagent available from Chemat. Available pack sizes: 10mg, 100mg, 2mg, 25mg, 5mg, 10mM (in 1ml dmso), 50mg. Offered by: GLPBio.

brandGLPBio
catalog numberGC12932-10
cas1380288-87-8
size10mg
Need more information?

Ask us about this product — we're happy to help.

Available pack sizes

brand size price
GLPBio 10mg 1252.31 Pln
GLPBio 100mg 5048.20 Pln
GLPBio 2mg 742.14 Pln
GLPBio 25mg 2015.23 Pln
GLPBio 5mg 962.12 Pln
GLPBio 10mM (in 1ml dmso) 1107.21 Pln
GLPBio 50mg 3424.06 Pln

properties

purityNo data
delivery timeTo be confirmed by Chemat

Pinometostat (EPZ-5676) is a potent DOT1L histone methyltransferase inhibitor.

Source: ChEBI

Identity
Molecular formulaC30H42N8O3
Molecular weight562.7 g/mol
IUPAC name(2R,3R,4S,5R)-2-(6-aminopurin-9-yl)-5-[[[3-[2-(6-tert-butyl-1H-benzimidazol-2-yl)ethyl]cyclobutyl]-propan-2-ylamino]methyl]oxolane-3,4-diol
InChIKeyLXFOLMYKSYSZQS-XKHGBIBOSA-N
SMILESCC(C)N(C[C@@H]1[C@H]([C@H]([C@@H](O1)N2C=NC3=C(N=CN=C32)N)O)O)C4CC(C4)CCC5=NC6=C(N5)C=C(C=C6)C(C)(C)C

Computed by PubChem (NCBI)

Synonyms: pinometostat, Pinometostat, trans-, Pinometostat [INN], Pinometostat anhydrous, Pinometostat (EPZ5676), trans-pinometostat, Pinometostat(EPZ5676), Pinometostat(EPZ5676)?, PINOMETOSTAT [WHO-DD], orb1226408
Isomers (same molecular formula)
6-ethyl-3-[4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]-5-[(3R)-1-prop-2-enoylpyrrolidin-3-yl]oxypyrazine-2-carboxamide C30H42N8O3

Also listed as

9-(5-Deoxy-5-((cis-3-(2-(6-(1,1-dimethylethyl)-1H-benzimidazol-2-yl)ethyl)cyclobutyl)(1-methylethyl)amino)-beta-D-ribofuranosyl)-9H-purin-6-amine TRC CAS 1380288-87-8
Pinometostat/ 97.56% (existing batch purity) TargetMol CAS 1380288-87-8
9-(5-Deoxy-5-((cis-3-(2-(6-(1,1-dimethylethyl)-1H-benzimidazol-2-yl)ethyl)cyclobutyl)(1-methylethyl)amino)-beta-D-ribofuranosyl)-9H- purin-6-amine Biosynth CAS 1380288-87-8
Pinometostat, 95% Thermo Scientific (Acros) CAS 1380288-87-8
Pinometostat 98% Ambeed CAS 1380288-87-8
(2R,3R,4S,5R)-2-(6-Amino-9H-purin-9-yl)-5-((((lr,3S)-3-(2-(5-(tert-butyl)-lH-benzo[d]imidazol2yl)ethyl)cyclobutyl)(isopropyl)amino)methyl)tetrahydrofuran-3,4-diol, 98%, 98% Chemat CAS 1380288-87-8
Pinometostat, 99.99% MedChemExpress CAS 1380288-87-8
Pinometostat (Standard) MedChemExpress CAS 1380288-87-8
(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-{[(propan-2-yl)[(1r,3s)-3-[2-(6-tert-butyl-1H-1,3-benzodiazol-2-yl)ethyl]cyclobutyl]amino]methyl}oxolane-3,4-diol, 98% Fluorochem CAS 1380288-87-8