Products 1380288-87-8

CAS 1380288-87-8 appears in our catalog under these names: 9-(5-Deoxy-5-((cis-3-(2-(6-(1,1-dimethylethyl)-1H-benzimidazol-2-yl)ethyl)cyclobutyl)(1-methylethyl)amino)-beta-D-ribofuranosyl)-9H-purin-6-amine, Pinometostat/ 97.56% (existing batch purity), EPZ5676, 9-(5-Deoxy-5-((cis-3-(2-(6-(1,1-dimethylethyl)-1H-benzimidazol-2-yl)ethyl)cyclobutyl)(1-methylethyl)amino)-beta-D-ribofuranosyl)-9H- purin-6-amine, Pinometostat, 95%. Offered by: TRC, TargetMol, GLPBio, Biosynth, Thermo Scientific (Acros). Available pack sizes: 100mg, 2mg, 5mg, 10mg, 25mg, 10mM (in 1ml dmso), 50mg, 250mg.

9-(5-Deoxy-5-((cis-3-(2-(6-(1,1-dimethylethyl)-1H-benzimidazol-2-yl)ethyl)cyclobutyl)(1-methylethyl)amino)-beta-D-ribofuranosyl)-9H-purin-6-amine
TRC
  • size: 100mg
  • Variants: 1
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Pinometostat/ 97.56% (existing batch purity)
TargetMol
  • size: 2mg, 5mg, 10mg
  • Variants: 3
from 412.42
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EPZ5676
GLPBio
  • size: 10mg, 100mg, 2mg, 25mg
  • Variants: 7
from 742.14
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9-(5-Deoxy-5-((cis-3-(2-(6-(1,1-dimethylethyl)-1H-benzimidazol-2-yl)ethyl)cyclobutyl)(1-methylethyl)amino)-beta-D-ribofuranosyl)-9H- purin-6-amine
Biosynth
  • size: 5mg, 10mg, 25mg
  • Variants: 3
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Pinometostat, 95%
Thermo Scientific (Acros)
  • size: 100MG
  • Variants: 1
from 2525.67
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Pinometostat 98%
Ambeed
  • size: 250mg, 1mg, 2mg, 5mg
  • Variants: 7
from 253.56
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(2R,3R,4S,5R)-2-(6-Amino-9H-purin-9-yl)-5-((((lr,3S)-3-(2-(5-(tert-butyl)-lH-benzo[d]imidazol2yl)ethyl)cyclobutyl)(isopropyl)amino)methyl)tetrahydrofuran-3,4-diol, 98%, 98%
Chemat
  • size: 10mg, 50mg, 100mg, 250mg
  • Variants: 4
from 592.40
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Pinometostat, 99.99%
MedChemExpress
  • size: 50 mg, 5 mg, 25 mg, 10 mg
  • Variants: 6
from 454.37
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Pinometostat (Standard)
MedChemExpress
  • size: 10 mg, 25 mg, 5 mg, 50 mg
  • Variants: 6
from 468.30
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(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-{[(propan-2-yl)[(1r,3s)-3-[2-(6-tert-butyl-1H-1,3-benzodiazol-2-yl)ethyl]cyclobutyl]amino]methyl}oxolane-3,4-diol, 98%
Fluorochem
  • size: 10mg, 50mg, 100mg
  • Variants: 3
from 1106.92
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Pinometostat (EPZ-5676) is a potent DOT1L histone methyltransferase inhibitor.

Source: ChEBI

Identity
Molecular formulaC30H42N8O3
Molecular weight562.7 g/mol
IUPAC name(2R,3R,4S,5R)-2-(6-aminopurin-9-yl)-5-[[[3-[2-(6-tert-butyl-1H-benzimidazol-2-yl)ethyl]cyclobutyl]-propan-2-ylamino]methyl]oxolane-3,4-diol
InChIKeyLXFOLMYKSYSZQS-XKHGBIBOSA-N
SMILESCC(C)N(C[C@@H]1[C@H]([C@H]([C@@H](O1)N2C=NC3=C(N=CN=C32)N)O)O)C4CC(C4)CCC5=NC6=C(N5)C=C(C=C6)C(C)(C)C

Computed by PubChem (NCBI)

Synonyms: pinometostat, Pinometostat, trans-, Pinometostat [INN], Pinometostat anhydrous, Pinometostat (EPZ5676), trans-pinometostat, Pinometostat(EPZ5676), Pinometostat(EPZ5676)?, PINOMETOSTAT [WHO-DD], orb1226408
Isomers (same molecular formula)
6-ethyl-3-[4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]-5-[(3R)-1-prop-2-enoylpyrrolidin-3-yl]oxypyrazine-2-carboxamide C30H42N8O3