Epoxomicin

cas: 134381-21-8 — see every product listed under this CAS number, including other names

Epoxomicin (CAS 134381-21-8) is a chemical reagent available from Chemat. Available pack sizes: 1mg, 20mg, 5mg, 10mM (in 1ml dmso), 10mg, 0,2mg, 25mg, 50UG. Offered by: GLPBio, Biosynth, Sigma-Aldrich.

brandGLPBio
catalog numberGC12494-1
cas134381-21-8
size1mg
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Available pack sizes

brand size price
GLPBio 1mg 896.59 Pln
GLPBio 20mg 4416.33 Pln
GLPBio 5mg 1725.04 Pln
GLPBio 10mM (in 1ml dmso) 1991.83 Pln
Biosynth 10mg price on request
Biosynth 0,2mg price on request
Biosynth 5mg price on request
Biosynth 25mg price on request
Sigma-Aldrich 50UG 1560.00 Pln

properties

purityNo data
delivery timeTo be confirmed by Chemat
Structural formula: {0} (CAS {1})

Epoxomicin is a tripeptide consisting of an Ile-Ile-Thr-NH2 sequence N-substituted on the threonamide amidic nitrogen with a (2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl group and with acetyl and methyl groups on the nitrogen of the isoleucine residue distal to the threonamide; a naturally occurring selective proteasome inhibitor with anti-inflammatory activity. It has a role as a proteasome inhibitor. It is a member of morpholines and a tripeptide.

Source: ChEBI

Identity
Molecular formulaC28H50N4O7
Molecular weight554.7 g/mol
IUPAC name(2S,3S)-2-[[(2S,3S)-2-[acetyl(methyl)amino]-3-methylpentanoyl]amino]-N-[(2S,3R)-3-hydroxy-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxobutan-2-yl]-3-methylpentanamide
InChIKeyDOGIDQKFVLKMLQ-JTHVHQAWSA-N
SMILESCC[C@H](C)[C@@H](C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)[C@]1(CO1)C)NC(=O)[C@H]([C@@H](C)CC)N(C)C(=O)C

Computed by PubChem (NCBI)

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