GSK126 98%
cas: 1346574-57-9 — see every product listed under this CAS number, including other names
GSK126 98% (CAS 1346574-57-9) is a chemical reagent available from Chemat. Available pack sizes: 1mg, 5mg, 50mg, 100mg, 250mg, 1g. Offered by: Ambeed.
| brand | Ambeed |
|---|---|
| catalog number | A114568-1mg |
| cas | 1346574-57-9 |
| size | 1mg |
Documents:
Safety Data Sheet (MSDS)
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Available pack sizes
| brand | size | price | |
|---|---|---|---|
| Ambeed | 1mg | 170.12 Pln | |
| Ambeed | 5mg | 286.94 Pln | |
| Ambeed | 50mg | 887.69 Pln | |
| Ambeed | 100mg | 1371.62 Pln | |
| Ambeed | 250mg | 2144.81 Pln | |
| Ambeed | 1g | 5465.62 Pln |
properties
| purity | 98% |
|---|---|
| delivery time | 1-2 weeks |
| ambeed catalog no. | A114568 |
GSK126 is a member of the class of methylindoles that is 1H-indole substituted by (2S)-butan-2-yl, methyl, N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]acetamide, and 6-(piperazin-1-yl)pyridin-3-yl groups at positions 1, 3, 4, and 6, respectively. It is a potent and highly selective inhibitor of EZH2 methyltransferase (IC50 = 9.9 nM). It has a role as an antiatherosclerotic agent, an EC 2.1.1.43 (enhancer of zeste homolog 2) inhibitor, an antineoplastic agent, an angiogenesis inhibitor, a neuroprotective agent and an anti-obesity agent. It is a secondary carboxamide, a member of pyridines, a pyridone, a methylindole and a N-arylpiperazine.
Source: ChEBI
| Molecular formula | C31H38N6O2 |
|---|---|
| Molecular weight | 526.7 g/mol |
| IUPAC name | 1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-methyl-6-(6-piperazin-1-yl-3-pyridinyl)indole-4-carboxamide |
| InChIKey | FKSFKBQGSFSOSM-QFIPXVFZSA-N |
| SMILES | CC[C@H](C)N1C=C(C2=C(C=C(C=C21)C3=CN=C(C=C3)N4CCNCC4)C(=O)NCC5=C(C=C(NC5=O)C)C)C |
Computed by PubChem (NCBI)