GSK2656157

cas: 1337532-29-2 — see every product listed under this CAS number, including other names

GSK2656157 (CAS 1337532-29-2) is a chemical reagent available from Chemat. Available pack sizes: 10mg, 100mg, 10mM (in 1ml dmso), 50mg. Offered by: GLPBio.

brandGLPBio
catalog numberGC11068-10
cas1337532-29-2
size10mg
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Available pack sizes

brand size price
GLPBio 10mg 826.38 Pln
GLPBio 100mg 2038.63 Pln
GLPBio 10mM (in 1ml dmso) 938.72 Pln
GLPBio 50mg 1313.16 Pln

properties

purityNo data
delivery timeTo be confirmed by Chemat
Structural formula: {0} (CAS {1})

GSK2656157 is a pyrrolopyrimidine that is 7-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine which has been substituted at position 5 by a 4-fluoro-2,3-dihydro-1H-indol-5-yl group, the nitrogen of which has been acylated by a (6-methylpyridin-2-yl)acetyl group. An orally bioavailable PERK inhibitor. It has a role as a PERK inhibitor, an EC 3.1.3.48 (protein-tyrosine-phosphatase) inhibitor and an antineoplastic agent. It is a tertiary carboxamide, a member of indoles, a member of methylpyridines, an organofluorine compound, a pyrrolopyrimidine and a biaryl.

Source: ChEBI

Identity
Molecular formulaC23H21FN6O
Molecular weight416.5 g/mol
IUPAC name1-[5-(4-amino-7-methylpyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-2,3-dihydroindol-1-yl]-2-(6-methyl-2-pyridinyl)ethanone
InChIKeyPRWSIEBRGXYXAJ-UHFFFAOYSA-N
SMILESCC1=NC(=CC=C1)CC(=O)N2CCC3=C2C=CC(=C3F)C4=CN(C5=NC=NC(=C45)N)C

Computed by PubChem (NCBI)

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