Products 87051-43-2

CAS 87051-43-2 appears in our catalog under these names: Ritanserin, Ritanserin/ 99.89% (existing batch purity), Ritanserin, 99.89% ,, 99.89% ,, Ritanserin, 99.78%, Ritanserin (Standard). Offered by: TRC, TargetMol, GLPBio, Biosynth, Chemat. Available pack sizes: 2,5g, 1mg, 2mg, 5mg, 10mg, 25mg, 50mg, 100mg.

Ritanserin
TRC, GLPBio, Biosynth
  • size: 2,5g, 10mg, 25mg, 5mg
  • Variants: 9
from 639.16
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Ritanserin/ 99.89% (existing batch purity)
TargetMol
  • size: 1mg, 2mg, 5mg, 10mg
  • Variants: 7
from 412.42
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Ritanserin, 99.89% ,, 99.89% ,
Chemat
  • size: 1mg, 5mg, 2mg, 10mg
  • Variants: 8
from 386.00
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Ritanserin, 99.78%
MedChemExpress
  • size: 10 mg, 100 mg, 5 mg, 10mM/1mL
  • Variants: 6
from 407.93
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Ritanserin (Standard)
MedChemExpress
  • size: 5 mg, 50 mg, 25 mg, 10 mg
  • Variants: 5
from 839.82
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Ritanserin, 97%
Fluorochem
  • size: 100mg
  • Variants: 1
from 5136.75
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Structural formula: {0} (CAS {1})

Ritanserin is a thiazolopyrimidine that is 5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one which is substituted at position 7 by a methyl group and at position 6 by a 2-{4-[bis(4-fluorophenyl)methylidene]piperidin-1-yl}ethyl group. A potent and long-acting seratonin (5-hydroxytryptamine, 5-HT) antagonist of the subtype 5-HT2 (Ki = 0.39 nM), it is used in the treatment of a variety of disorders including anxiety, depression and schizophrenia. It has little sedative action. It has a role as an antidepressant, an anxiolytic drug, an antipsychotic agent, a serotonergic antagonist, a dopaminergic antagonist and an EC 3.4.21.26 (prolyl oligopeptidase) inhibitor. It is a member of piperidines, an organofluorine compound and a thiazolopyrimidine.

Source: ChEBI

Identity
Molecular formulaC27H25F2N3OS
Molecular weight477.6 g/mol
IUPAC name6-[2-[4-[bis(4-fluorophenyl)methylidene]piperidin-1-yl]ethyl]-7-methyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
InChIKeyJUQLTPCYUFPYKE-UHFFFAOYSA-N
SMILESCC1=C(C(=O)N2C=CSC2=N1)CCN3CCC(=C(C4=CC=C(C=C4)F)C5=CC=C(C=C5)F)CC3

Computed by PubChem (NCBI)

Synonyms: ritanserin, Tiserton, Ritanserina, Ritanserine, Ritanserinum, Ritanserine [French], Ritanserinum [Latin], Ritanserina [Spanish], Ritanserin [USAN:INN:BAN], Ritanserin, powder