SB-224289 Hyrochloride

cas: 180084-26-8 — see every product listed under this CAS number, including other names

SB-224289 Hyrochloride (CAS 180084-26-8) is a chemical reagent available from Chemat. Available pack sizes: 25mg, 50mg, 100mg. Offered by: Biosynth.

brandBiosynth
catalog numberFHA08426-25mg
cas180084-26-8
size25mg
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Available pack sizes

brand size price
Biosynth 25mg price on request
Biosynth 50mg price on request
Biosynth 100mg price on request

properties

categoryLife Sciences
purityNo data
delivery time3-4 Weeks
Structural formula: {0} (CAS {1})

SB 224289 hydrochloride is a hydrochloride that is the monohydrochloride salt of SB 224289. Selective 5-HT1B receptor antagonist (pKi = 8.2). Displays >60-fold selectivity over 5-HT1D, 5-HT1A, 5-HT1E, 5-HT1F, 5-HT2A and 5-HT2C receptors in radioligand binding and functional assays. Centrally active following oral administration in vivo. It has a role as a serotonergic antagonist and a prodrug. It contains a SB 224289(1+).

Source: ChEBI

Identity
Molecular formulaC32H33ClN4O3
Molecular weight557.1 g/mol
IUPAC name[4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]phenyl]-(1'-methylspiro[6,7-dihydro-2H-furo[2,3-f]indole-3,4'-piperidine]-5-yl)methanone;hydrochloride
InChIKeyGKGKBZYMDILCOF-UHFFFAOYSA-N
SMILESCC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)N4CCC5=CC6=C(C=C54)C7(CCN(CC7)C)CO6.Cl

Computed by PubChem (NCBI)

Also listed as