Products 519055-62-0

CAS 519055-62-0 appears in our catalog under these names: Tasisulam, Tasisulam/ 99.97% (existing batch purity), Tasisulam, >95.0%(HPLC)(qNMR), Tasisulam 95%, N-((5-Bromothiophen-2-yl)sulfonyl)-2,4-dichlorobenzamide, 95%, 95%. Offered by: GLPBio, TargetMol, TCI, Ambeed, Chemat. Available pack sizes: 10mg, 10mM (in 1ml dmso), 50mg, 5mg, 25mg, 100mg, 200mg, 500mg.

Tasisulam
GLPBio
  • size: 10mg, 10mM (in 1ml dmso), 50mg
  • Variants: 3
from 667.25
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Tasisulam/ 99.97% (existing batch purity)
TargetMol
  • size: 5mg, 10mg, 25mg, 50mg
  • Variants: 7
from 419.13
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Tasisulam, >95.0%(HPLC)(qNMR)
TCI
  • size: 10mg
  • Variants: 1
from 580.57
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Tasisulam 95%
Ambeed
  • size: 1mg, 5mg, 10mg, 25mg
  • Variants: 8
from 159.00
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N-((5-Bromothiophen-2-yl)sulfonyl)-2,4-dichlorobenzamide, 95%, 95%
Chemat
  • size: 1mg, 5mg, 10mg, 25mg
  • Variants: 5
from 136.40
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Tasisulam, 99.77%
MedChemExpress
  • size: 100 mg, 10 mg, 10mM/1mL, 5 mg
  • Variants: 6
from 342.91
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Tasisulam, 95%
Fluorochem
  • size: 5mg, 10mg, 25mg, 250mg
  • Variants: 4
from 258.26
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Structural formula: {0} (CAS {1})

Tasisulam is a thiophene substituted by a 2,4-dichlorobenzamide-N-sulfonyl and bromo groups at positions 2 and 4, respectively. It induces tumour cell apoptosis via ROS induction and mitochondrial membrane potential loss and currently in clinical development for the treatment of cancer. It has a role as an antineoplastic agent, an angiogenesis inhibitor and an apoptosis inducer. It is a dichlorobenzene, a member of thiophenes, an organobromine compound and a N-sulfonylcarboxamide.

Source: ChEBI

Identity
Molecular formulaC11H6BrCl2NO3S2
Molecular weight415.1 g/mol
IUPAC nameN-(5-bromothiophen-2-yl)sulfonyl-2,4-dichlorobenzamide
InChIKeyWWONFUQGBVOKOF-UHFFFAOYSA-N
SMILESC1=CC(=C(C=C1Cl)Cl)C(=O)NS(=O)(=O)C2=CC=C(S2)Br

Computed by PubChem (NCBI)

Synonyms: Tasisulam, N-(2,4-Dichlorobenzoyl)-5-bromothiophene-2-sulfonamide, N-[(5-bromothiophen-2-yl)sulfonyl]-2,4-dichlorobenzamide, tasisulamum, Tasisulam [INN], N-(5-bromothiophen-2-yl)sulfonyl-2,4-dichlorobenzamide, Tasisulam (sodium), Tasisulam(LY573636), N-(5-bromothiophen-2-ylsulfonyl)-2,4-dichlorobenzamide, N-[(5-bromo-2-thienyl)sulfonyl]-2,4-dichloro-benzamide