Products 210101-16-9

CAS 210101-16-9 appears in our catalog under these names: Conivaptan, 98%, Conivaptan. Offered by: Chemat Brand, Biosynth, MedChemExpress. Available pack sizes: on request, 50mg, 25mg, 100mg, 500mg, 250mg, Get quote.

Conivaptan, 98%
Chemat Brand
  • size: on request
  • Variants: 1
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Conivaptan
Biosynth, MedChemExpress
  • size: 50mg, 25mg, 100mg, 500mg
  • Variants: 6
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Conivaptan is the amide resulting from the formal condensation of 4-[(biphenyl-2-ylcarbonyl)amino]benzoic acid with the benzazepine nitrogen of 2-methyl-1,4,5,6-tetrahydroimidazo[4,5-d][1]benzazepine. It is an antagonist for two of the three types of arginine vasopressin (AVP) receptors, V1a and V2. It is used as its hydrochloride salt for the treatment of hyponatraemia (low blood sodium levels) caused by syndrome of inappropriate antidiuretic hormone (SIADH). It has a role as an aquaretic and a vasopressin receptor antagonist.

Source: ChEBI

Identity
Molecular formulaC32H26N4O2
Molecular weight498.6 g/mol
IUPAC nameN-[4-(2-methyl-4,5-dihydro-3H-imidazo[4,5-d][1]benzazepine-6-carbonyl)phenyl]-2-phenylbenzamide
InChIKeyIKENVDNFQMCRTR-UHFFFAOYSA-N
SMILESCC1=NC2=C(N1)CCN(C3=CC=CC=C32)C(=O)C4=CC=C(C=C4)NC(=O)C5=CC=CC=C5C6=CC=CC=C6

Computed by PubChem (NCBI)

Synonyms: Conivaptan, conivaptanum, Conivaptan [INN], Conivaptan (INN), CONIVAPTAN [MI], CONIVAPTAN [VANDF], CONIVAPTAN [WHO-DD], IKENVDNFQMCRTR-UHFFFAOYSA-N
Related forms of this compound
2-phenyl-N-[2,3,5,6-tetradeuterio-4-(2-methyl-4,5-dihydro-3H-imidazo[4,5-d][1]benzazepine-6-carbonyl)phenyl]benzamide C32H26N4O2