Crenigacestat, 99.01%
cas: 1421438-81-4 — see every product listed under this CAS number, including other names
Crenigacestat, 99.01% (CAS 1421438-81-4) is a chemical reagent available from Chemat. Available pack sizes: 10mM/1mL, 1 mg, 10 mg, 100 mg, 25 mg, 50 mg, 5 mg. Offered by: MedChemExpress.
| brand | MedChemExpress |
|---|---|
| catalog number | HY-12449-10mM/1mL |
| cas | 1421438-81-4 |
| size | 10mM/1mL |
| availability | In stock |
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Available pack sizes
| brand | size | price | |
|---|---|---|---|
| MedChemExpress | 10mM/1mL | 853.75 Pln | |
| MedChemExpress | 1 mg | 459.01 Pln | |
| MedChemExpress | 10 mg | 1318.15 Pln | |
| MedChemExpress | 100 mg | 6115.40 Pln | |
| MedChemExpress | 25 mg | 2279.46 Pln | |
| MedChemExpress | 50 mg | 3719.10 Pln | |
| MedChemExpress | 5 mg | 839.82 Pln |
properties
| delivery time | 1-2 weeks |
|---|---|
| purity | 99.01% |
Crenigacestat (LY3039478) is an orally active Notch and g-secretase inhibitor, with an IC50 of 1 nM in most of the tumor cell lines tested.
Source: ChEBI
| Molecular formula | C22H23F3N4O4 |
|---|---|
| Molecular weight | 464.4 g/mol |
| IUPAC name | 4,4,4-trifluoro-N-[(2S)-1-[[(7S)-5-(2-hydroxyethyl)-6-oxo-7H-pyrido[2,3-d][3]benzazepin-7-yl]amino]-1-oxopropan-2-yl]butanamide |
| InChIKey | YCBAQKQAINQRFW-UGSOOPFHSA-N |
| SMILES | C[C@@H](C(=O)N[C@H]1C2=CC=CC=C2C3=C(N=CC=C3)N(C1=O)CCO)NC(=O)CCC(F)(F)F |
Computed by PubChem (NCBI)