GBR 12909 dihydrochloride

cas: 67469-78-7 — see every product listed under this CAS number, including other names

GBR 12909 dihydrochloride (CAS 67469-78-7) is a chemical reagent available from Chemat. Available pack sizes: 50mg, 100mg, 250mg, 500mg. Offered by: Biosynth.

brandBiosynth
catalog numberFG65030-50mg
cas67469-78-7
size50mg
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Available pack sizes

brand size price
Biosynth 50mg price on request
Biosynth 100mg price on request
Biosynth 250mg price on request
Biosynth 500mg price on request

properties

categoryLife Sciences
sub-category 1Ligands
sub-category 2Transporters
purityNo data
delivery time1-2 weeks

Vanoxerine dihydrochloride is a hydrochloride salt that is obtained by reaction of vanoxerine with two equivalents of hydrogen chloride. Potent, competitive inhibitor of dopamine uptake (Ki = 1 nM for inhibition of striatal dopamine uptake). Has > 100-fold lower affinity for the noradrenalin and 5-HT uptake carriers. Also a potent sigma ligand (IC50 = 48 nM). Centrally active following systemic administration. It has a role as a dopamine uptake inhibitor. It contains a vanoxerine(2+).

Source: ChEBI

Identity
Molecular formulaC28H34Cl2F2N2O
Molecular weight523.5 g/mol
IUPAC name1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine;dihydrochloride
InChIKeyMIBSKSYCRFWIRU-UHFFFAOYSA-N
SMILESC1CN(CCN1CCCC2=CC=CC=C2)CCOC(C3=CC=C(C=C3)F)C4=CC=C(C=C4)F.Cl.Cl

Computed by PubChem (NCBI)

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