GI 254023X
cas: 260264-93-5 — see every product listed under this CAS number, including other names
GI 254023X (CAS 260264-93-5) is a chemical reagent available from Chemat. Available pack sizes: 500mg, 1mg, 2mg, 5mg, 25mg, 10mg. Offered by: TRC, GLPBio, Biosynth.
| brand | TRC |
|---|---|
| catalog number | TRC-G377200-500MG |
| cas | 260264-93-5 |
| size | 500mg |
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Available pack sizes
| brand | size | price | |
|---|---|---|---|
| TRC | 500mg | price on request | |
| GLPBio | 1mg | 976.16 Pln | |
| Biosynth | 1mg | price on request | |
| Biosynth | 2mg | price on request | |
| Biosynth | 5mg | price on request | |
| Biosynth | 25mg | price on request | |
| Biosynth | 10mg | price on request |
properties
| purity | No data |
|---|---|
| delivery time | To be confirmed by Chemat |
GI254023X is a L-valine derivative that is 3-methyl-L-valine in which carboxy OH group is replaced by a methylnitrilo group and the one of the amino hydrogens is replaced by a (2R)-2-{(1S)-1-[formyl(hydroxy)amino]ethyl}-5-phenylpentanoyl group. It is a potent MMP9 and ADAM10 metalloprotease inhibitor with IC50 of 2.5 and 5.3 nM, respectively. It has a role as an antineoplastic agent, a matrix metalloproteinase inhibitor, an EC 3.4.24.* (metalloendopeptidase) inhibitor and an apoptosis inducer. It is an aldehyde, a member of hydroxylamines and a L-valine derivative.
Source: ChEBI
| Molecular formula | C21H33N3O4 |
|---|---|
| Molecular weight | 391.5 g/mol |
| IUPAC name | (2R)-N-[(2S)-3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide |
| InChIKey | GHVMTHKJUAOZJP-CGTJXYLNSA-N |
| SMILES | C[C@@H]([C@@H](CCCC1=CC=CC=C1)C(=O)N[C@H](C(=O)NC)C(C)(C)C)N(C=O)O |
Computed by PubChem (NCBI)