GI254023X, 99.67%
cas: 260264-93-5 — see every product listed under this CAS number, including other names
GI254023X, 99.67% (CAS 260264-93-5) is a chemical reagent available from Chemat. Available pack sizes: 1 mg, 50 mg, 5 mg, 10 mg, 25 mg, 100 mg, 10mM/1mL. Offered by: MedChemExpress.
| brand | MedChemExpress |
|---|---|
| catalog number | HY-19956-1 mg |
| cas | 260264-93-5 |
| size | 1 mg |
| availability | Get quote |
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Available pack sizes
| brand | size | price | |
|---|---|---|---|
| MedChemExpress | 1 mg | 811.96 Pln | |
| MedChemExpress | 50 mg | 4099.91 Pln | |
| MedChemExpress | 5 mg | 1081.31 Pln | |
| MedChemExpress | 10 mg | 1559.64 Pln | |
| MedChemExpress | 25 mg | 2613.83 Pln | |
| MedChemExpress | 100 mg | 5878.56 Pln | |
| MedChemExpress | 10mM/1mL | 1294.93 Pln |
properties
| delivery time | over 3 weeks |
|---|---|
| purity | 99.67% |
GI254023X is a L-valine derivative that is 3-methyl-L-valine in which carboxy OH group is replaced by a methylnitrilo group and the one of the amino hydrogens is replaced by a (2R)-2-{(1S)-1-[formyl(hydroxy)amino]ethyl}-5-phenylpentanoyl group. It is a potent MMP9 and ADAM10 metalloprotease inhibitor with IC50 of 2.5 and 5.3 nM, respectively. It has a role as an antineoplastic agent, a matrix metalloproteinase inhibitor, an EC 3.4.24.* (metalloendopeptidase) inhibitor and an apoptosis inducer. It is an aldehyde, a member of hydroxylamines and a L-valine derivative.
Source: ChEBI
| Molecular formula | C21H33N3O4 |
|---|---|
| Molecular weight | 391.5 g/mol |
| IUPAC name | (2R)-N-[(2S)-3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide |
| InChIKey | GHVMTHKJUAOZJP-CGTJXYLNSA-N |
| SMILES | C[C@@H]([C@@H](CCCC1=CC=CC=C1)C(=O)N[C@H](C(=O)NC)C(C)(C)C)N(C=O)O |
Computed by PubChem (NCBI)