GR 127935 hydrochloride hydrate

cas: 148642-42-6 — see every product listed under this CAS number, including other names

GR 127935 hydrochloride hydrate (CAS 148642-42-6) is a chemical reagent available from Chemat. Available pack sizes: 250mg, 25mg, 50mg, 100mg, 500mg, 10MG. Offered by: Biosynth, Sigma-Aldrich.

brandBiosynth
catalog numberBG177433-250mg
cas148642-42-6
size250mg
Need more information?

Ask us about this product — we're happy to help.

Available pack sizes

brand size price
Biosynth 250mg price on request
Biosynth 25mg price on request
Biosynth 50mg price on request
Biosynth 100mg price on request
Biosynth 500mg price on request
Sigma-Aldrich 10MG 1080.00 Pln

properties

categoryLife Sciences
purityNo data
delivery time3-4 Weeks

GR 127935 hydrochloride is a hydrochloride obtained by reaction of GR 127935 with one equivalent of hydrochloric acid. Potent and selective 5-HT1B/1D receptor antagonist (pKi values are 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors). Displays > 100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other receptor types. Centrally active following oral administration. It has a role as a serotonergic antagonist. It contains a GR 127935(1+).

Source: ChEBI

Identity
Molecular formulaC29H32ClN5O3
Molecular weight534.0 g/mol
IUPAC nameN-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide;hydrochloride
InChIKeySRVVUYIJVBLEJI-UHFFFAOYSA-N
SMILESCC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)NC4=CC(=C(C=C4)OC)N5CCN(CC5)C.Cl

Computed by PubChem (NCBI)

Synonyms: C29H32ClN5O3, orb1704510, Tox21_500790

Also listed as

GR 127935 Hydrochloride Hydrate, >95% (HPLC) TRC CAS 148642-42-6
GR 127935 hydrochloride TargetMol CAS 148642-42-6
GR 127935 hydrochloride GLPBio CAS 148642-42-6
GR 127935 hydrochloride, 98%, 98% Chemat CAS 148642-42-6
GR127935 (hydrochloride), 99.38% MedChemExpress CAS 148642-42-6