GR 127935 hydrochloride

cas: 148642-42-6 — see every product listed under this CAS number, including other names

GR 127935 hydrochloride (CAS 148642-42-6) is a chemical reagent available from Chemat. Available pack sizes: 5mg, 10mg, 25mg, 50mg. Offered by: TargetMol, GLPBio.

brandTargetMol
catalog numberT22806-5mg
cas148642-42-6
size5mg
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Available pack sizes

brand size price
TargetMol 5mg 1899.92 Pln
TargetMol 10mg 3241.52 Pln
TargetMol 25mg 6382.54 Pln
TargetMol 50mg 11934.53 Pln
GLPBio 10mg 1533.14 Pln
GLPBio 25mg 2745.39 Pln
GLPBio 5mg 1037.01 Pln
GLPBio 50mg 4772.05 Pln

properties

purityNo data
delivery timeon request

GR 127935 hydrochloride is a hydrochloride obtained by reaction of GR 127935 with one equivalent of hydrochloric acid. Potent and selective 5-HT1B/1D receptor antagonist (pKi values are 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors). Displays > 100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other receptor types. Centrally active following oral administration. It has a role as a serotonergic antagonist. It contains a GR 127935(1+).

Source: ChEBI

Identity
Molecular formulaC29H32ClN5O3
Molecular weight534.0 g/mol
IUPAC nameN-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide;hydrochloride
InChIKeySRVVUYIJVBLEJI-UHFFFAOYSA-N
SMILESCC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)NC4=CC(=C(C=C4)OC)N5CCN(CC5)C.Cl

Computed by PubChem (NCBI)

Synonyms: C29H32ClN5O3, orb1704510, Tox21_500790

Also listed as

GR 127935 Hydrochloride Hydrate, >95% (HPLC) TRC CAS 148642-42-6
GR 127935 hydrochloride GLPBio CAS 148642-42-6
GR 127935 hydrochloride hydrate Biosynth CAS 148642-42-6
GR 127935 hydrochloride, 98%, 98% Chemat CAS 148642-42-6
GR127935 (hydrochloride), 99.38% MedChemExpress CAS 148642-42-6