Galunisertib, 99.95%

cas: 700874-72-2 — see every product listed under this CAS number, including other names

Galunisertib, 99.95% (CAS 700874-72-2) is a chemical reagent available from Chemat. Available pack sizes: 500 mg, 50 mg, 5 mg, 1 g, 10mM/1mL, 10 mg, 100 mg, 200 mg. Offered by: MedChemExpress.

brand	MedChemExpress
catalog number	HY-13226-500 mg
cas	700874-72-2
size	500 mg
availability	In stock

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Available pack sizes

brand	size	price
MedChemExpress	500 mg	3719.10 Pln
MedChemExpress	50 mg	839.82 Pln
MedChemExpress	5 mg	361.49 Pln
MedChemExpress	1 g	5516.33 Pln
MedChemExpress	10mM/1mL	384.71 Pln
MedChemExpress	10 mg	454.37 Pln
MedChemExpress	100 mg	1318.15 Pln
MedChemExpress	200 mg	1917.23 Pln

properties

delivery time	1-2 weeks
purity	99.95%

LY-2157299 is a pyrrolopyrazole that is 5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole which is substituted at positions 2 and 3 by 6-methylpyridin-2-yl and 6-(aminocarbonyl)quinolin-4-yl groups, respectively. A Transforming growth factor-betaRI (TGF-betaRI) kinase inhibitor, it blocks TGF-beta-mediated tumor growth in glioblastoma. It has a role as an antineoplastic agent and a TGFbeta receptor antagonist. It is a member of methylpyridines, a member of quinolines, a monocarboxylic acid amide, a pyrrolopyrazole and an aromatic amide.

Source: ChEBI

Identity
Molecular formula	C₂₂H₁₉N₅O
Molecular weight	369.4 g/mol
IUPAC name	4-[2-(6-methyl-2-pyridinyl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]quinoline-6-carboxamide
InChIKey	IVRXNBXKWIJUQB-UHFFFAOYSA-N
SMILES	CC1=NC(=CC=C1)C2=NN3CCCC3=C2C4=C5C=C(C=CC5=NC=C4)C(=O)N

Computed by PubChem (NCBI)

Synonyms: Galunisertib, galunisertibum, Galunisertib (LY2157299), ly2157299(galunisertib), Galunisertib [USAN], Galunisertib [USAN:INN], Galunisertib (USAN/INN), GALUNISERTIB [INN], GALUNISERTIB [WHO-DD], orb1224194