Rimonabant (Standard)
cas: 168273-06-1 — see every product listed under this CAS number, including other names
Rimonabant (Standard) (CAS 168273-06-1) is a chemical reagent available from Chemat. Available pack sizes: 100 mg, 5 mg, 50 mg, 25 mg, 10 mg. Offered by: MedChemExpress.
| brand | MedChemExpress |
|---|---|
| catalog number | HY-14136R-100 mg |
| cas | 168273-06-1 |
| size | 100 mg |
| availability | Get quote |
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Available pack sizes
| brand | size | price | |
|---|---|---|---|
| MedChemExpress | 100 mg | 2883.18 Pln | |
| MedChemExpress | 5 mg | 505.45 Pln | |
| MedChemExpress | 50 mg | 1963.67 Pln | |
| MedChemExpress | 25 mg | 1346.02 Pln | |
| MedChemExpress | 10 mg | 733.01 Pln |
properties
| delivery time | over 3 weeks |
|---|---|
| purity | no data |
Rimonabant is a carbohydrazide obtained by formal condensation of the carboxy group of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid with the amino group of 1-aminopiperidine. It is a potent and selective cannabinoid receptor 1 (CB1R) antagonist. Besides its antagonistic properties, numerous studies have shown that, at micromolar concentrations rimonabant behaves as an inverse agonist at CB1 receptors. The drug was the first selective CB1 antagonist/inverse agonist introduced into clinical practice to treat obesity and metabolic-related disorders. It was later withdrawn from market due to CNS-related adverse effects including depression and suicidal ideation. It has a role as an appetite depressant, a CB1 receptor antagonist and an anti-obesity agent. It is a dichlorobenzene, a member of pyrazoles, a carbohydrazide, an amidopiperidine and a member of monochlorobenzenes.
Source: ChEBI
| Molecular formula | C22H21Cl3N4O |
|---|---|
| Molecular weight | 463.8 g/mol |
| IUPAC name | 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide |
| InChIKey | JZCPYUJPEARBJL-UHFFFAOYSA-N |
| SMILES | CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)Cl |
Computed by PubChem (NCBI)