CAS 179248-59-0 appears in our catalog under these names: Src Inhibitor 1/ 100%, Src I1, Src Inhibitor 1, Src Inhibitor 1 99%, Src Inhibitor 1, 99.97%. Offered by: TargetMol, GLPBio, Biosynth, Ambeed, MedChemExpress. Available pack sizes: 1mg, 2mg, 5mg, 10mg, 25mg, 50mg, 100mg, 500mg.
Src Inhibitor-1 is a member of the class of quinazolines that is quinazoline which is substituted at position 4 by a p-phenoxyanilino group and at positions 6 and 7 by methoxy groups. It is a potent, competitive dual site (both the ATP- and peptide-binding) Src kinase inhibitor. Src Inhibitor-1 is one of the 'gold standards' for Src kinase inhibition that has been shown to use PP1 or PP2 in parallel with Src-I1 to inhbit Src family kinases. It has a role as an EC 2.7.10.2 (non-specific protein-tyrosine kinase) inhibitor. It is an aromatic ether, a member of quinazolines, a polyether and a secondary amino compound.
Source: ChEBI
| Molecular formula | C22H19N3O3 |
|---|---|
| Molecular weight | 373.4 g/mol |
| IUPAC name | 6,7-dimethoxy-N-(4-phenoxyphenyl)quinazolin-4-amine |
| InChIKey | DMWVGXGXHPOEPT-UHFFFAOYSA-N |
| SMILES | COC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=C(C=C3)OC4=CC=CC=C4)OC |
Computed by PubChem (NCBI)