AZD2858 99%

cas: 486424-20-8 — see every product listed under this CAS number, including other names

AZD2858 99% (CAS 486424-20-8) is a chemical reagent available from Chemat. Available pack sizes: 1mg, 5mg, 10mg, 50mg, 100mg, 250mg. Offered by: Ambeed.

brandAmbeed
catalog numberA128237-1mg
cas486424-20-8
size1mg
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Available pack sizes

brand size price
Ambeed 1mg 264.69 Pln
Ambeed 5mg 420.44 Pln
Ambeed 10mg 620.69 Pln
Ambeed 50mg 1049.00 Pln
Ambeed 100mg 1727.62 Pln
Ambeed 250mg 2884.62 Pln

properties

purity99%
delivery time 2-3 weeks
ambeed catalog no.A128237
Structural formula: {0} (CAS {1})

AZD2858 is a member of the class of pyrazines that is pyrazine substituted by (pyridin-3-yl)aminocarbonyl, amino, and 4-(4-methylpiperazine-1-sulfonyl)phenyl groups at positions 2, 3 and 6, respectively. It is a potent inhibitor of GSK3alpha and GSK3beta (IC50 values of 0.9 and 4.9 nM, respectively) and increases bone mass (via Wnt activation) in rats. It has a role as a Wnt signalling activator, an antineoplastic agent, a bone density conservation agent and an EC 2.7.11.26 (tau-protein kinase) inhibitor. It is a secondary carboxamide, a member of pyridines, an aromatic amine, a sulfonamide, a member of pyrazines and a N-methylpiperazine.

Source: ChEBI

Identity
Molecular formulaC21H23N7O3S
Molecular weight453.5 g/mol
IUPAC name3-amino-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]-N-pyridin-3-ylpyrazine-2-carboxamide
InChIKeyFHCSBLWRGCOVPT-UHFFFAOYSA-N
SMILESCN1CCN(CC1)S(=O)(=O)C2=CC=C(C=C2)C3=CN=C(C(=N3)C(=O)NC4=CN=CC=C4)N

Computed by PubChem (NCBI)

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