MK-2461, 99.28%
cas: 917879-39-1 — see every product listed under this CAS number, including other names
MK-2461, 99.28% (CAS 917879-39-1) is a chemical reagent available from Chemat. Available pack sizes: 10 mg, 100 mg, 25 mg, 10mM/1mL, 5 mg, 50 mg. Offered by: MedChemExpress.
| brand | MedChemExpress |
|---|---|
| catalog number | HY-50703-10 mg |
| cas | 917879-39-1 |
| size | 10 mg |
| availability | In stock |
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Available pack sizes
| brand | size | price | |
|---|---|---|---|
| MedChemExpress | 10 mg | 1285.64 Pln | |
| MedChemExpress | 100 mg | 5256.26 Pln | |
| MedChemExpress | 25 mg | 2339.83 Pln | |
| MedChemExpress | 10mM/1mL | 914.12 Pln | |
| MedChemExpress | 5 mg | 849.11 Pln | |
| MedChemExpress | 50 mg | 3496.19 Pln |
properties
| delivery time | 1-2 weeks |
|---|---|
| purity | 99.28% |
MK-2461 is a member of the class of benzocycloheptapyridines that is 5H-benzo[4,5]cyclohepta[1,2-b]pyridin-5-one substituted by 1-methyl-1H-pyrazol-4-yl and [{[(2R)-1,4-dioxan-2-yl]methyl}(methyl)sulfamoyl]amino groups at positions 3 and 7, respectively. It is a novel ATP-competitive multi-targeted inhibitor of activated c-Met (IC50 = 2.5 nM). It has a role as an antineoplastic agent, an apoptosis inducer and a c-Met tyrosine kinase inhibitor. It is a member of pyrazoles, a member of dioxanes, a benzocycloheptapyridine and a member of sulfamides.
Source: ChEBI
| Molecular formula | C24H25N5O5S |
|---|---|
| Molecular weight | 495.6 g/mol |
| IUPAC name | 14-[[[(2R)-1,4-dioxan-2-yl]methyl-methylsulfamoyl]amino]-5-(1-methylpyrazol-4-yl)-2-oxo-7-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,9,12,14-heptaene |
| InChIKey | JGEBLDKNWBUGRZ-HXUWFJFHSA-N |
| SMILES | CN1C=C(C=N1)C2=CC3=C(C=CC4=C(C3=O)C=C(C=C4)NS(=O)(=O)N(C)C[C@@H]5COCCO5)N=C2 |
Computed by PubChem (NCBI)