Rigosertib-d6
cas: 592542-59-1 — see every product listed under this CAS number, including other names
Rigosertib-d6 (CAS 592542-59-1) is a chemical reagent available from Chemat. Available pack sizes: 50mg, 100mg. Offered by: Biosynth.
| brand | Biosynth |
|---|---|
| catalog number | SYA54259-50mg |
| cas | 592542-59-1 |
| size | 50mg |
Need more information?
Ask us about this product — we're happy to help.
Available pack sizes
| brand | size | price | |
|---|---|---|---|
| Biosynth | 50mg | price on request | |
| Biosynth | 100mg | price on request |
properties
| category | Life Sciences |
|---|---|
| purity | No data |
| delivery time | 3-4 Weeks |
Rigosertib is an N-[2-methoxy-5-({[2-(2,4,6-trimethoxyphenyl)ethenyl]sulfonyl}methyl)phenyl]glycine in which the double bond has E-configuration. It is a non-ATP-competitive inhibitor of PLK1 with an IC50 of 9 nM and exhibits anti-cancer properties. It has a role as an EC 2.7.11.21 (polo kinase) inhibitor, an antineoplastic agent, a microtubule-destabilising agent and an apoptosis inducer. It is a conjugate acid of a rigosertib(1-).
Source: ChEBI
| Molecular formula | C21H25NO8S |
|---|---|
| Molecular weight | 451.5 g/mol |
| IUPAC name | 2-[2-methoxy-5-[[(E)-2-(2,4,6-trimethoxyphenyl)ethenyl]sulfonylmethyl]anilino]acetic acid |
| InChIKey | OWBFCJROIKNMGD-BQYQJAHWSA-N |
| SMILES | COC1=C(C=C(C=C1)CS(=O)(=O)/C=C/C2=C(C=C(C=C2OC)OC)OC)NCC(=O)O |
Computed by PubChem (NCBI)