MK 4827

cas: 1038915-60-4 — see every product listed under this CAS number, including other names

MK 4827 (CAS 1038915-60-4) is a chemical reagent available from Chemat. Available pack sizes: 0,025g, 0,05g, 0,1g, 0,25g, 0,5g. Offered by: Biosynth.

brandBiosynth
catalog numberFP35532-0,025g
cas1038915-60-4
size0,025g
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Available pack sizes

brand size price
Biosynth 0,025g price on request
Biosynth 0,05g price on request
Biosynth 0,1g price on request
Biosynth 0,25g price on request
Biosynth 0,5g price on request

properties

categoryLife Sciences
sub-category 1Ligands
sub-category 2Enzyme Modulators
purityNo data
delivery time1-2 weeks

Niraparib is a 2-[4-(piperidin-3-yl)phenyl]-2H-indazole-7-carboxamide that has S-configuration. It is a potent inhibitor of PARP1 and PARP2 (IC50 of 3.8 and 2.1 nM, respectively) and approved as a first-line maintenance treatment for women with advanced ovarian cancer after responding to platinum-based chemotherapy. It has a role as a radiosensitizing agent, an antineoplastic agent, an EC 2.4.2.30 (NAD(+) ADP-ribosyltransferase) inhibitor and an apoptosis inducer.

Source: ChEBI

Identity
Molecular formulaC19H20N4O
Molecular weight320.4 g/mol
IUPAC name2-[4-[(3S)-piperidin-3-yl]phenyl]indazole-7-carboxamide
InChIKeyPCHKPVIQAHNQLW-CQSZACIVSA-N
SMILESC1C[C@H](CNC1)C2=CC=C(C=C2)N3C=C4C=CC=C(C4=N3)C(=O)N

Computed by PubChem (NCBI)

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