MK–4827

cas: 1038915-60-4 — see every product listed under this CAS number, including other names

MK–4827 (CAS 1038915-60-4) is a chemical reagent available from Chemat. Available pack sizes: 10mg, 100mg, 5mg, 50mg. Offered by: GLPBio.

brandGLPBio
catalog numberGC17802-10
cas1038915-60-4
size10mg
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Available pack sizes

brand size price
GLPBio 10mg 859.15 Pln
GLPBio 100mg 2899.85 Pln
GLPBio 5mg 676.61 Pln
GLPBio 50mg 2141.60 Pln

properties

purityNo data
delivery timeTo be confirmed by Chemat

Niraparib is a 2-[4-(piperidin-3-yl)phenyl]-2H-indazole-7-carboxamide that has S-configuration. It is a potent inhibitor of PARP1 and PARP2 (IC50 of 3.8 and 2.1 nM, respectively) and approved as a first-line maintenance treatment for women with advanced ovarian cancer after responding to platinum-based chemotherapy. It has a role as a radiosensitizing agent, an antineoplastic agent, an EC 2.4.2.30 (NAD(+) ADP-ribosyltransferase) inhibitor and an apoptosis inducer.

Source: ChEBI

Identity
Molecular formulaC19H20N4O
Molecular weight320.4 g/mol
IUPAC name2-[4-[(3S)-piperidin-3-yl]phenyl]indazole-7-carboxamide
InChIKeyPCHKPVIQAHNQLW-CQSZACIVSA-N
SMILESC1C[C@H](CNC1)C2=CC=C(C=C2)N3C=C4C=CC=C(C4=N3)C(=O)N

Computed by PubChem (NCBI)

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